Mitoxantrone dihydrochloride;鹽酸米托蒽醌;70476-82-3
僅用于工業應用或科學研究,不可用于人類或動物的臨床診斷或治療,非藥用.Mitoxantrone dihydrochloride is a potent topoisomerase II inhibitor. Mitoxantrone dihydrochloride also inhibits protein kinase C (PKC) activity with an IC50 of 8.5 μM. Mitoxantrone dihydrochloride induces apoptosis of B-CLL (B-chronic lymphocytic leukaemia) cells. Mitoxantrone dihydrochloride shows antitumor activity.Mitoxantrone dihydrochloride 是一種有效的拓撲異構酶II (topoisomerase II) 抑制劑。Mitoxantrone dihydrochloride 也可抑制蛋白激酶 C (PKC),其 IC50 值為 8.5 μM。Mitoxantrone dihydrochloride 誘導 B- 慢性淋巴細胞白血病 (B-CLL) 細胞凋亡 (apoptosis)